Clinical data
Fazadon
Identifiers
(E)-bis(3-methyl-2-phenylimidazo[3,2-a]
pyridin-4-ium-1-yl)diazene dibromide
PubChem CID
CompTox Dashboard (EPA)
Chemical and physical data
C28H24Br2N6
604.350 g·mol−1
3D model (JSmol)
Cc1c(n(c2[n+]1cccc2)N=Nn3c4cccc[n+]4c(c3c5ccccc5)C)c6ccccc6.[Br-].[Br-]
InChI=1S/C28H24N6.2BrH/c1-21-27(23-13-5-3-6-14-23)33(25-17-9-11-19-31(21)25)29-30-34-26-18-10-12-20-32(26)22(2)28(34)24-15-7-4-8-16-24;;/h3-20H,1-2H3;2*1H/q+2;;/p-2 N
Key:LBOZSXSPRGACHC-UHFFFAOYSA-L N
Fazadinium bromide is a muscle relaxant which acts as a nicotinic acetylcholine receptor antagonist through neuromuscular blockade.[1]
Peripherally acting
(primarily antinicotinic,
NMJ block)
Other
nAChRsTooltip Nicotinic acetylcholine receptors
Antagonists
(and NAMsTooltip negative allosteric modulators)
Precursors
(and prodrugs)
This drug article relating to the musculoskeletal system is a stub. You can help Wikipedia by expanding it.