Receptor (ligands) |
GlyRTooltip Glycine receptor |
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Positive modulators: Alcohols (e.g., brometone, chlorobutanol (chloretone), ethanol (alcohol), tert-butanol (2M2P), tribromoethanol, trichloroethanol, trifluoroethanol)
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Alkylbenzene sulfonate
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Anandamide
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Barbiturates (e.g., pentobarbital, sodium thiopental)
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Chlormethiazole
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D12-116
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Dihydropyridines (e.g., nicardipine)
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Etomidate
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Ginseng constituents (e.g., ginsenosides (e.g., ginsenoside-Rf))
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Glutamic acid (glutamate)
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Ivermectin
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Ketamine
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Neuroactive steroids (e.g., alfaxolone, pregnenolone (eltanolone), pregnenolone acetate, minaxolone, ORG-20599)
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Nitrous oxide
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Penicillin G
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Propofol
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Tamoxifen
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Tetrahydrocannabinol
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Triclofos
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Tropeines (e.g., atropine, bemesetron, cocaine, LY-278584, tropisetron, zatosetron)
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Volatiles/gases (e.g., chloral hydrate, chloroform, desflurane, diethyl ether (ether), enflurane, halothane, isoflurane, methoxyflurane, sevoflurane, toluene, trichloroethane (methyl chloroform), trichloroethylene)
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Xenon
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Zinc
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Antagonists: 2-Aminostrychnine
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2-Nitrostrychnine
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4-Phenyl-4-formyl-N-methylpiperidine
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αEMBTL
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Bicuculline
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Brucine
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Cacotheline
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Caffeine
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Colchicine
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Colubrine
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Cyanotriphenylborate
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Dendrobine
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Diaboline
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Endocannabinoids (e.g., 2-AG, anandamide (AEA))
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Gaboxadol (THIP)
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Gelsemine
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iso-THAZ
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Isobutyric acid
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Isonipecotic acid
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Isostrychnine
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Laudanosine
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N-Methylbicuculline
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N-Methylstrychnine
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N,N-Dimethylmuscimol
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Nipecotic acid
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Pitrazepin
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Pseudostrychnine
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Quinolines (e.g., 4-hydroxyquinoline, 4-hydroxyquinoline-3-carboxylic acid, 5,7-CIQA, 7-CIQ, 7-TFQ, 7-TFQA)
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RU-5135
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Sinomenine
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Strychnine
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Thiocolchicoside
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Tutin
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Negative modulators: Amiloride
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Benzodiazepines (e.g., bromazepam, clonazepam, diazepam, flunitrazepam, flurazepam)
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Corymine
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Cyanotriphenylborate
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Daidzein
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Dihydropyridines (e.g., nicardipine, nifedipine, nitrendipine)
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Furosemide
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Genistein
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Ginkgo constituents (e.g., bilobalide, ginkgolides (e.g., ginkgolide A, ginkgolide B, ginkgolide C, ginkgolide J, ginkgolide M))
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Imipramine
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NBQX
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Neuroactive steroids (e.g., 3α-androsterone sulfate, 3β-androsterone sulfate, deoxycorticosterone, DHEA sulfate, pregnenolone sulfate, progesterone)
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Opioids (e.g., codeine, dextromethorphan, dextrorphan, levomethadone, levorphanol, morphine, oripavine, pethidine, thebaine)
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Picrotoxin (i.e., picrotin and picrotoxinin)
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PMBA
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Riluzole
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Tropeines (e.g., bemesetron, LY-278584, tropisetron, zatosetron)
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Verapamil
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Zinc
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NMDARTooltip N-Methyl-D-aspartate receptor |
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