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Chemical and physical data | |
Formula | C8H10ClN3S |
Molar mass | 215.70 g/mol g·mol−1 |
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Tiamenidine is a compound that shares many of the pharmacological properties of clonidine.
Reaction of thiourea 1 with methyl iodide gives the corresponding S-methyl analogue (2), followed by heating with ethylenediamine, completes the synthesis of Tiamenidine (3).
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Sympatholytics (antagonize α-adrenergic vasoconstriction) |
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Other antagonists |
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α1 |
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α2 |
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β |
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