t
e
|
---|
α1 |
Agonists |
|
---|
Antagonists |
-
Abanoquil
-
Ajmalicine
-
Alfuzosin
-
Anisodamine
-
Anisodine
-
Atiprosin
-
Atypical antipsychotics (e.g., brexpiprazole, clozapine, olanzapine, quetiapine, risperidone)
-
Benoxathian
-
Beta blockers (e.g., adimolol, amosulalol, arotinolol, carvedilol, eugenodilol, labetalol)
-
Buflomedil
-
Bunazosin
-
Corynanthine
-
Dapiprazole
-
Domesticine
-
Doxazosin
-
Ergolines (e.g., acetergamine, ergotamine, dihydroergotamine, lisuride, nicergoline, terguride)
-
Etoperidone
-
Fenspiride
-
Hydroxyzine
-
Indoramin
-
Ketanserin
-
L-765,314
-
mCPP
-
Mepiprazole
-
Metazosin
-
Monatepil
-
Moxisylyte
-
Naftopidil
-
Nantenine
-
Neldazosin
-
Niaprazine
-
Niguldipine
-
Pardoprunox
-
Pelanserin
-
Perlapine
-
Phendioxan
-
Phenoxybenzamine
-
Phentolamine
-
Phenylpiperazine antidepressants (e.g., hydroxynefazodone, nefazodone, trazodone, triazoledione)
-
Piperoxan
-
Prazosin
-
Quinazosin
-
Quinidine
-
Silodosin
-
Spegatrine
-
Spiperone
-
Talipexole
-
Tamsulosin
-
Terazosin
-
Tiodazosin
-
Tolazoline
-
Tetracyclic antidepressants (e.g., amoxapine, maprotiline, mianserin)
-
Tricyclic antidepressants (e.g., amitriptyline, clomipramine, doxepin, imipramine, trimipramine)
-
Trimazosin
-
Typical antipsychotics (e.g., chlorpromazine, fluphenazine, loxapine, thioridazine)
-
Urapidil
-
WB-4101
-
Zolertine
|
---|
|
---|
α2 |
Agonists |
|
---|
Antagonists |
-
1-PP
-
Adimolol
-
Amesergide
-
Aptazapine
-
Atipamezole
-
Atypical antipsychotics (e.g., asenapine, brexpiprazole, clozapine, lurasidone, olanzapine, paliperidone, quetiapine, risperidone, zotepine)
-
Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone)
-
BRL-44408
-
Buflomedil
-
Cirazoline
-
Efaroxan
-
Esmirtazapine
-
Fenmetozole
-
Fluparoxan
-
Idazoxan
-
Ketanserin
-
Lisuride
-
mCPP
-
Mianserin
-
Mirtazapine
-
NAN-190
-
Pardoprunox
-
Phentolamine
-
Phenoxybenzamine
-
Piperoxan
-
Piribedil
-
Rauwolscine
-
Rotigotine
-
Setiptiline
-
Spegatrine
-
Spiroxatrine
-
Sunepitron
-
Terguride
-
Tolazoline
-
Typical antipsychotics (e.g., chlorpromazine, fluphenazine, loxapine, thioridazine)
-
Yohimbine
|
---|
|
---|
β |
|
---|
|
t
e
|
---|
Alcohols |
|
---|
Barbiturates |
|
---|
Benzodiazepines |
|
---|
Carbamates |
|
---|
Flavonoids |
|
---|
Imidazoles |
|
---|
Kava constituents |
|
---|
Monoureides |
|
---|
Neuroactive steroids |
|
---|
Nonbenzodiazepines |
|
---|
Phenols |
|
---|
Piperidinediones |
|
---|
Pyrazolopyridines |
|
---|
Quinazolinones |
|
---|
Volatiles/gases |
|
---|
Others/unsorted |
-
3-Hydroxybutanal
-
α-EMTBL
-
AA-29504
-
Alogabat
-
Avermectins (e.g., ivermectin)
-
Bromide compounds (e.g., lithium bromide, potassium bromide, sodium bromide)
-
Carbamazepine
-
Chloralose
-
Chlormezanone
-
Clomethiazole
-
Darigabat
-
DEABL
-
Deuterated etifoxine
-
Dihydroergolines (e.g., dihydroergocryptine, dihydroergosine, dihydroergotamine, ergoloid (dihydroergotoxine))
-
DS2
-
Efavirenz
-
Etazepine
-
Etifoxine
-
Fenamates (e.g., flufenamic acid, mefenamic acid, niflumic acid, tolfenamic acid)
-
Fluoxetine
-
Flupirtine
-
Hopantenic acid
-
KRM-II-81
-
Lanthanum
-
Lavender oil
-
Lignans (e.g., 4-O-methylhonokiol, honokiol, magnolol, obovatol)
-
Loreclezole
-
Menthyl isovalerate (validolum)
-
Monastrol
-
Niacin
-
Niacinamide
-
Org 25,435
-
Phenytoin
-
Propanidid
-
Retigabine (ezogabine)
-
Safranal
-
Seproxetine
-
Stiripentol
-
Sulfonylalkanes (e.g., sulfonmethane (sulfonal), tetronal, trional)
-
Terpenoids (e.g., borneol)
-
Topiramate
-
Valerian constituents (e.g., isovaleric acid, isovaleramide, valerenic acid, valerenol)
|
---|
See also: Receptor/signaling modulators • GABA receptor modulators • GABA metabolism/transport modulators
|
t
e
|
---|
H1 |
Agonists |
|
---|
Antagonists |
-
Others: Atypical antipsychotics (e.g., aripiprazole, asenapine, brexpiprazole, brilaroxazine, clozapine, iloperidone, olanzapine, paliperidone, quetiapine, risperidone, ziprasidone, zotepine)
-
Phenylpiperazine antidepressants (e.g., hydroxynefazodone, nefazodone, trazodone, triazoledione)
-
Tetracyclic antidepressants (e.g., amoxapine, loxapine, maprotiline, mianserin, mirtazapine, oxaprotiline)
-
Tricyclic antidepressants (e.g., amitriptyline, butriptyline, clomipramine, desipramine, dosulepin (dothiepin), doxepin, imipramine, iprindole, lofepramine, nortriptyline, protriptyline, trimipramine)
-
Typical antipsychotics (e.g., chlorpromazine, flupenthixol, fluphenazine, loxapine, perphenazine, prochlorperazine, thioridazine, thiothixene)
|
---|
|
---|
H2 |
|
---|
H3 |
|
---|
H4 |
|
---|
-
See also
-
Receptor/signaling modulators
-
Monoamine metabolism modulators
-
Monoamine reuptake inhibitors
|
t
e
|
---|
DATTooltip Dopamine transporter (DRIsTooltip Dopamine reuptake inhibitors) |
|
---|
NETTooltip Norepinephrine transporter (NRIsTooltip Norepinephrine reuptake inhibitors) |
|
|
|
|
|
|
-
Others: Antihistamines (e.g., brompheniramine, chlorphenamine, pheniramine, tripelennamine)
-
Antipsychotics (e.g., loxapine, ziprasidone)
-
Arylcyclohexylamines (e.g., ketamine, phencyclidine)
-
Dopexamine
-
Ephenidine
-
Ginkgo biloba
-
Indeloxazine
-
Nefazodone
-
Opioids (e.g., desmetramadol, methadone, pethidine (meperidine), tapentadol, tramadol, levorphanol)
|
|
---|
SERTTooltip Serotonin transporter (SRIsTooltip Serotonin reuptake inhibitors) |
|
|
|
|
-
Others: A-80426
-
Amoxapine
-
Antihistamines (e.g., brompheniramine, chlorphenamine, dimenhydrinate, diphenhydramine, mepyramine (pyrilamine), pheniramine, tripelennamine)
-
Antipsychotics (e.g., loxapine, ziprasidone)
-
Arylcyclohexylamines (e.g., 3-MeO-PCP, esketamine, ketamine, methoxetamine, phencyclidine)
-
Cyclobenzaprine
-
Delucemine
-
Dextromethorphan
-
Dextrorphan
-
Efavirenz
-
Hypidone
-
Medifoxamine
-
Mesembrine
-
Mifepristone
-
MIN-117 (WF-516)
-
N-Me-5-HT
-
Opioids (e.g., dextropropoxyphene, methadone, pethidine (meperidine), levorphanol, tapentadol, tramadol)
-
Roxindole
|
|
---|
VMATsTooltip Vesicular monoamine transporters |
|
---|
Others |
|
---|
See also: Receptor/signaling modulators • Monoamine releasing agents • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins
|
t
e
|
---|
mAChRsTooltip Muscarinic acetylcholine receptors |
Agonists |
|
---|
Antagonists |
-
3-Quinuclidinyl benzilate
-
4-DAMP
-
Aclidinium bromide (+formoterol)
-
Abediterol
-
AF-DX 250
-
AF-DX 384
-
Ambutonium bromide
-
Anisodamine
-
Anisodine
-
Antihistamines (first-generation) (e.g., brompheniramine, buclizine, captodiame, chlorphenamine (chlorpheniramine), cinnarizine, clemastine, cyproheptadine, dimenhydrinate, dimetindene, diphenhydramine, doxylamine, meclizine, mequitazine, perlapine, phenindamine, pheniramine, phenyltoloxamine, promethazine, propiomazine, triprolidine)
-
AQ-RA 741
-
Atropine
-
Atropine methonitrate
-
Atypical antipsychotics (e.g., clozapine, fluperlapine, olanzapine (+fluoxetine), rilapine, quetiapine, tenilapine, zotepine)
-
Benactyzine
-
Benzatropine (benztropine)
-
Benzilone
-
Benzilylcholine mustard
-
Benzydamine
-
Bevonium
-
BIBN 99
-
Biperiden
-
Bornaprine
-
Camylofin
-
CAR-226,086
-
CAR-301,060
-
CAR-302,196
-
CAR-302,282
-
CAR-302,368
-
CAR-302,537
-
CAR-302,668
-
Caramiphen
-
Cimetropium bromide
-
Clidinium bromide
-
Cloperastine
-
CS-27349
-
Cyclobenzaprine
-
Cyclopentolate
-
Darifenacin
-
DAU-5884
-
Desfesoterodine
-
Dexetimide
-
DIBD
-
Dicycloverine (dicyclomine)
-
Dihexyverine
-
Difemerine
-
Diphemanil metilsulfate
-
Ditran
-
Drofenine
-
EA-3167
-
EA-3443
-
EA-3580
-
EA-3834
-
Emepronium bromide
-
Etanautine
-
Etybenzatropine (ethybenztropine)
-
Fenpiverinium
-
Fentonium bromide
-
Fesoterodine
-
Flavoxate
-
Glycopyrronium bromide (+beclometasone/formoterol, +indacaterol, +neostigmine)
-
Hexahydrodifenidol
-
Hexahydrosiladifenidol
-
Hexbutinol
-
Hexocyclium
-
Himbacine
-
HL-031,120
-
Homatropine
-
Imidafenacin
-
Ipratropium bromide (+salbutamol)
-
Isopropamide
-
J-104,129
-
Hyoscyamine
-
Mamba toxin 3
-
Mamba toxin 7
-
Mazaticol
-
Mebeverine
-
Meladrazine
-
Mepenzolate
-
Methantheline
-
Methoctramine
-
Methylatropine
-
Methylhomatropine
-
Methylscopolamine
-
Metixene
-
Muscarinic toxin 7
-
N-Ethyl-3-piperidyl benzilate
-
N-Methyl-3-piperidyl benzilate
-
Nefopam
-
Octatropine methylbromide (anisotropine methylbromide)
-
Orphenadrine
-
Otenzepad (AF-DX 116)
-
Otilonium bromide
-
Oxapium iodide
-
Oxitropium bromide
-
Oxybutynin
-
Oxyphencyclimine
-
Oxyphenonium bromide
-
PBID
-
PD-102,807
-
PD-0298029
-
Penthienate
-
Pethidine
-
pFHHSiD
-
Phenglutarimide
-
Phenyltoloxamine
-
Pipenzolate bromide
-
Piperidolate
-
Pirenzepine
-
Piroheptine
-
Pizotifen
-
Poldine
-
Pridinol
-
Prifinium bromide
-
Procyclidine
-
Profenamine (ethopropazine)
-
Propantheline bromide
-
Propiverine
-
Quinidine
-
3-Quinuclidinyl thiochromane-4-carboxylate
-
Revefenacin
-
Rociverine
-
RU-47,213
-
SCH-57,790
-
SCH-72,788
-
SCH-217,443
-
Scopolamine (hyoscine)
-
Scopolamine butylbromide (hyoscine butylbromide)
-
Silahexacyclium
-
Sofpironium bromide
-
Solifenacin
-
SSRIsTooltip Selective serotonin reuptake inhibitors (e.g., femoxetine, paroxetine)
-
Telenzepine
-
Terodiline
-
Tetracyclic antidepressants (e.g., amoxapine, maprotiline, mianserin, mirtazapine)
-
Tiemonium iodide
-
Timepidium bromide
-
Tiotropium bromide
-
Tiquizium bromide
-
Tofenacin
-
Tolterodine
-
Tricyclic antidepressants (e.g., amitriptyline (+perphenazine), amitriptylinoxide, butriptyline, cidoxepin, clomipramine, desipramine, desmethyldesipramine, dibenzepin, dosulepin (dothiepin), doxepin, imipramine, lofepramine, nitroxazepine, northiaden (desmethyldosulepin), nortriptyline, protriptyline, quinupramine, trimipramine)
-
Tridihexethyl
-
Trihexyphenidyl
-
Trimebutine
-
Tripitamine (tripitramine)
-
Tropacine
-
Tropatepine
-
Tropicamide
-
Trospium chloride
-
Typical antipsychotics (e.g., chlorpromazine, chlorprothixene, cyamemazine (cyamepromazine), loxapine, mesoridazine, thioridazine)
-
Umeclidinium bromide (+vilanterol)
-
WIN-2299
-
Xanomeline
-
Zamifenacin
|
---|
|
---|
Precursors (and prodrugs) |
|
---|
-
See also
-
Receptor/signaling modulators
-
Nicotinic acetylcholine receptor modulators
-
Acetylcholine metabolism/transport modulators
|
t
e
|
---|
5-HT1 |
5-HT1A |
-
Agonists: 8-OH-DPAT
-
Adatanserin
-
Amphetamine
-
Antidepressants (e.g., etoperidone, hydroxynefazodone, nefazodone, trazodone, triazoledione, vilazodone, vortioxetine)
-
Atypical antipsychotics (e.g., aripiprazole, asenapine, brexpiprazole, cariprazine, clozapine, lurasidone, quetiapine, ziprasidone)
-
Azapirones (e.g., buspirone, eptapirone, gepirone, perospirone, tandospirone)
-
Bay R 1531
-
Befiradol
-
BMY-14802
-
Cannabidiol
-
Dimemebfe
-
Dopamine
-
Ebalzotan
-
Eltoprazine
-
Enciprazine
-
Ergolines (e.g., bromocriptine, cabergoline, dihydroergotamine, ergotamine, lisuride, LSD, methylergometrine (methylergonovine), methysergide, pergolide)
-
F-11,461
-
F-12826
-
F-13714
-
F-14679
-
F-15063
-
F-15,599
-
Flesinoxan
-
Flibanserin
-
Flumexadol
-
Hypidone
-
Lesopitron
-
LY-293284
-
LY-301317
-
mCPP
-
MKC-242
-
Naluzotan
-
NBUMP
-
Osemozotan
-
Oxaflozane
-
Pardoprunox
-
Piclozotan
-
Rauwolscine
-
Repinotan
-
Roxindole
-
RU-24,969
-
S-14,506
-
S-14671
-
S-15535
-
Sarizotan
-
Serotonin (5-HT)
-
SSR-181507
-
Sunepitron
-
Tryptamines (e.g., 5-CT, 5-MeO-DMT, 5-MT, bufotenin, DMT, indorenate, N-Me-5-HT, psilocin, psilocybin)
-
TGBA01AD
-
U-92,016-A
-
Urapidil
-
Vilazodone
-
Xaliproden
-
Yohimbine
|
-
Antagonists: Atypical antipsychotics (e.g., iloperidone, risperidone, sertindole)
-
AV965
-
Beta blockers (e.g., alprenolol, carteolol, cyanopindolol, iodocyanopindolol, isamoltane, oxprenolol, penbutolol, pindobind, pindolol, propranolol, tertatolol)
-
BMY-7,378
-
CSP-2503
-
Dotarizine
-
Ergolines (e.g., metergoline)
-
FCE-24379
-
Flopropione
-
GR-46611
-
Isamoltane
-
Lecozotan
-
Mefway
-
Metitepine (methiothepin)
-
MIN-117 (WF-516)
-
MPPF
-
NAN-190
-
Robalzotan
-
S-15535
-
SB-649,915
-
SDZ 216-525
-
Spiperone
-
Spiramide
-
Spiroxatrine
-
UH-301
-
WAY-100135
-
WAY-100635
-
Xylamidine
|
|
|
---|
5-HT1B |
-
Agonists: Anpirtoline
-
CGS-12066A
-
CP-93129
-
CP-94253
-
CP-122,288
-
CP-135807
-
Eltoprazine
-
Ergolines (e.g., bromocriptine, dihydroergotamine, ergotamine, methylergometrine (methylergonovine), methysergide, pergolide)
-
mCPP
-
RU-24,969
-
Serotonin (5-HT)
-
Triptans (e.g., avitriptan, donitriptan, eletriptan, sumatriptan, zolmitriptan)
-
TFMPP
-
Tryptamines (e.g., 5-BT, 5-CT, 5-MT, DMT)
-
Vortioxetine
|
|
|
|
---|
5-HT1D |
-
Agonists: CP-122,288
-
CP-135807
-
CP-286601
-
Ergolines (e.g., bromocriptine, cabergoline, dihydroergotamine, ergotamine, LSD, methysergide)
-
GR-46611
-
L-694247
-
L-772405
-
mCPP
-
PNU-109291
-
PNU-142633
-
Serotonin (5-HT)
-
TGBA01AD
-
Triptans (e.g., almotriptan, avitriptan, donitriptan, eletriptan, frovatriptan, naratriptan, rizatriptan, sumatriptan, zolmitriptan)
-
Tryptamines (e.g., 5-BT, 5-CT, 5-Et-DMT, 5-MT, 5-(nonyloxy)tryptamine, DMT)
|
|
|
|
---|
5-HT1E |
|
---|
5-HT1F |
|
---|
|
---|
5-HT2 |
5-HT2A |
-
Agonists: 25H/NB series (e.g., 25I-NBF, 25I-NBMD, 25I-NBOH, 25I-NBOMe, 25B-NBOMe, 25C-NBOMe, 25TFM-NBOMe, 2CBCB-NBOMe, 25CN-NBOH, 2CBFly-NBOMe)
-
2Cs (e.g., 2C-B, 2C-E, 2C-I, 2C-T-2, 2C-T-7, 2C-T-21)
-
2C-B-FLY
-
2CB-Ind
-
5-Methoxytryptamines (5-MeO-DET, 5-MeO-DiPT, 5-MeO-DMT, 5-MeO-DPT, 5-MT)
-
α-Alkyltryptamines (e.g., 5-Cl-αMT, 5-Fl-αMT, 5-MeO-αET, 5-MeO-αMT, α-Me-5-HT, αET, αMT)
-
AL-34662
-
AL-37350A
-
Bromo-DragonFLY
-
Dimemebfe
-
DMBMPP
-
DOx (e.g., DOB, DOC, DOI, DOM)
-
Efavirenz
-
Ergolines (e.g., 1P-LSD, ALD-52, bromocriptine, cabergoline, ergine (LSA), ergometrine (ergonovine), ergotamine, lisuride, LA-SS-Az, LSB, LSD, LSD-Pip, LSH, LSP, methylergometrine (methylergonovine), pergolide)
-
Flumexadol
-
IHCH-7113
-
Jimscaline
-
Lorcaserin
-
MDxx (e.g., MDA (tenamfetamine), MDMA (midomafetamine), MDOH, MMDA)
-
O-4310
-
Oxaflozane
-
PHA-57378
-
PNU-22394
-
PNU-181731
-
RH-34
-
SCHEMBL5334361
-
Phenethylamines (e.g., lophophine, mescaline)
-
Piperazines (e.g., BZP, quipazine, TFMPP)
-
Serotonin (5-HT)
-
TCB-2
-
TFMFly
-
Tryptamines (e.g., 5-BT, 5-CT, bufotenin, DET, DiPT, DMT, DPT, psilocin, psilocybin, tryptamine)
|
-
Antagonists: 5-I-R91150
-
5-MeO-NBpBrT
-
AC-90179
-
Adatanserin
-
Altanserin
-
Antihistamines (e.g., cyproheptadine, hydroxyzine, ketotifen, perlapine)
-
AMDA
-
Atypical antipsychotics (e.g., amperozide, aripiprazole, asenapine, blonanserin, brexpiprazole, carpipramine, clocapramine, clorotepine, clozapine, fluperlapine, gevotroline, iloperidone, lurasidone, melperone, mosapramine, ocaperidone, olanzapine, paliperidone, quetiapine, risperidone, sertindole, zicronapine, ziprasidone, zotepine)
-
Chlorprothixene
-
Cinanserin
-
CSP-2503
-
Deramciclane
-
Dotarizine
-
Eplivanserin
-
Ergolines (e.g., amesergide, LY-53857, LY-215,840, mesulergine, metergoline, methysergide, sergolexole)
-
Fananserin
-
Flibanserin
-
Glemanserin
-
Irindalone
-
Ketanserin
-
KML-010
-
Landipirdine
-
LY-393558
-
mCPP
-
Medifoxamine
-
Metitepine (methiothepin)
-
MIN-117 (WF-516)
-
Naftidrofuryl
-
Nantenine
-
Nelotanserin
-
Opiranserin (VVZ-149)
-
Pelanserin
-
Phenoxybenzamine
-
Pimavanserin
-
Pirenperone
-
Pizotifen
-
Pruvanserin
-
Rauwolscine
-
Ritanserin
-
Roluperidone
-
S-14671
-
Sarpogrelate
-
Serotonin antagonists and reuptake inhibitors (e.g., etoperidone, hydroxynefazodone, lubazodone, mepiprazole, nefazodone, triazoledione, trazodone)
-
SR-46349B
-
TGBA01AD
-
Teniloxazine
-
Temanogrel
-
Tetracyclic antidepressants (e.g., amoxapine, aptazapine, esmirtazapine, maprotiline, mianserin, mirtazapine)
-
Tricyclic antidepressants (e.g., amitriptyline)
-
Typical antipsychotics (e.g., chlorpromazine, fluphenazine, haloperidol, loxapine, perphenazine, pimozide, pipamperone, prochlorperazine, setoperone, spiperone, spiramide, thioridazine, thiothixene, trifluoperazine)
-
Volinanserin
-
Xylamidine
-
Yohimbine
|
|
|
---|
5-HT2B |
-
Agonists: 4-Methylaminorex
-
Aminorex
-
Amphetamines (e.g., chlorphentermine, cloforex, dexfenfluramine, fenfluramine, levofenfluramine, norfenfluramine)
-
BW-723C86
-
DOx (e.g., DOB, DOC, DOI, DOM)
-
Ergolines (e.g., cabergoline, dihydroergocryptine, dihydroergotamine, ergotamine, methylergometrine (methylergonovine), methysergide, pergolide)
-
Lorcaserin
-
MDxx (e.g., MDA (tenamfetamine), MDMA (midomafetamine), MDOH, MMDA)
-
Piperazines (e.g., TFMPP)
-
PNU-22394
-
Ro60-0175
-
Serotonin (5-HT)
-
Tryptamines (e.g., 5-BT, 5-CT, 5-MT, α-Me-5-HT, bufotenin, DET, DiPT, DMT, DPT, psilocin, psilocybin, tryptamine)
|
-
Antagonists: Agomelatine
-
Atypical antipsychotics (e.g., amisulpride, aripiprazole, asenapine, brexpiprazole, cariprazine, clozapine, N-desalkylquetiapine (norquetiapine), N-desmethylclozapine (norclozapine), olanzapine, pipamperone, quetiapine, risperidone, ziprasidone)
-
Cyproheptadine
-
EGIS-7625
-
Ergolines (e.g., amesergide, bromocriptine, lisuride, LY-53857, LY-272015, mesulergine)
-
Ketanserin
-
LY-393558
-
mCPP
-
Metadoxine
-
Metitepine (methiothepin)
-
Pirenperone
-
Pizotifen
-
Propranolol
-
PRX-08066
-
Rauwolscine
-
Ritanserin
-
RS-127445
-
Sarpogrelate
-
SB-200646
-
SB-204741
-
SB-206553
-
SB-215505
-
SB-221284
-
SB-228357
-
SDZ SER-082
-
Tegaserod
-
Tetracyclic antidepressants (e.g., amoxapine, mianserin, mirtazapine)
-
Trazodone
-
Typical antipsychotics (e.g., chlorpromazine)
-
TIK-301
-
Yohimbine
|
|
|
---|
5-HT2C |
-
Agonists: 2Cs (e.g., 2C-B, 2C-E, 2C-I, 2C-T-2, 2C-T-7, 2C-T-21)
-
5-Methoxytryptamines (5-MeO-DET, 5-MeO-DiPT, 5-MeO-DMT, 5-MeO-DPT, 5-MT)
-
α-Alkyltryptamines (e.g., 5-Cl-αMT, 5-Fl-αMT, 5-MeO-αET, 5-MeO-αMT, α-Me-5-HT, αET, αMT)
-
A-372159
-
AL-38022A
-
Alstonine
-
CP-809101
-
Dimemebfe
-
DOx (e.g., DOB, DOC, DOI, DOM)
-
Ergolines (e.g., ALD-52, cabergoline, dihydroergotamine, ergine (LSA), ergotamine, lisuride, LA-SS-Az, LSB, LSD, LSD-Pip, LSH, LSP, pergolide)
-
Flumexadol
-
Lorcaserin
-
MDxx (e.g., MDA (tenamfetamine), MDMA (midomafetamine), MDOH, MMDA)
-
MK-212
-
ORG-12962
-
ORG-37684
-
Oxaflozane
-
PHA-57378
-
Phenethylamines (e.g., lophophine, mescaline)
-
Piperazines (e.g., aripiprazole, BZP, mCPP, quipazine, TFMPP)
-
PNU-22394
-
PNU-181731
-
Ro60-0175
-
Ro60-0213
-
Serotonin (5-HT)
-
Tryptamines (e.g., 5-BT, 5-CT, bufotenin, DET, DiPT, DMT, DPT, psilocin, psilocybin, tryptamine)
-
Vabicaserin
-
WAY-629
-
WAY-161503
-
YM-348
|
-
Antagonists: Adatanserin
-
Agomelatine
-
Atypical antipsychotics (e.g., asenapine, clorotepine, clozapine, fluperlapine, iloperidone, melperone, olanzapine, paliperidone, quetiapine, risperidone, sertindole, ziprasidone, zotepine)
-
Captodiame
-
CEPC
-
Cinanserin
-
Cyproheptadine
-
Deramciclane
-
Desmetramadol
-
Dotarizine
-
Eltoprazine
-
Ergolines (e.g., amesergide, bromocriptine, LY-53857, LY-215,840, mesulergine, metergoline, methysergide, sergolexole)
-
Etoperidone
-
Fluoxetine
-
FR-260010
-
Irindalone
-
Ketanserin
-
Ketotifen
-
Latrepirdine (dimebolin)
-
Medifoxamine
-
Metitepine (methiothepin)
-
Nefazodone
-
Pirenperone
-
Pizotifen
-
Propranolol
-
Ritanserin
-
RS-102221
-
S-14671
-
SB-200646
-
SB-206553
-
SB-221284
-
SB-228357
-
SB-242084
-
SB-243213
-
SDZ SER-082
-
Tedatioxetine
-
Tetracyclic antidepressants (e.g., amoxapine, aptazapine, esmirtazapine, maprotiline, mianserin, mirtazapine)
-
TIK-301
-
Tramadol
-
Trazodone
-
Tricyclic antidepressants (e.g., amitriptyline, nortriptyline)
-
Typical antipsychotics (e.g., chlorpromazine, loxapine, pimozide, pipamperone, thioridazine)
-
Xylamidine
|
|
|
---|
|
---|
5-HT3–7 |
5-HT3 |
-
Agonists: Alcohols (e.g., butanol, ethanol (alcohol), trichloroethanol)
-
m-CPBG
-
Phenylbiguanide
-
Piperazines (e.g., BZP, mCPP, quipazine)
-
RS-56812
-
Serotonin (5-HT)
-
SR-57227
-
SR-57227A
-
Tryptamines (e.g., 2-Me-5-HT, 5-CT, bufotenidine (5-HTQ))
-
Volatiles/gases (e.g., halothane, isoflurane, toluene, trichloroethane)
-
YM-31636
|
-
Antagonists: Alosetron
-
Anpirtoline
-
Arazasetron
-
AS-8112
-
Atypical antipsychotics (e.g., clozapine, olanzapine, quetiapine)
-
Azasetron
-
Batanopride
-
Bemesetron (MDL-72222)
-
Bupropion
-
Cilansetron
-
CSP-2503
-
Dazopride
-
Dolasetron
-
Galanolactone
-
Granisetron
-
Hydroxybupropion
-
Lerisetron
-
Memantine
-
Ondansetron
-
Palonosetron
-
Ramosetron
-
Renzapride
-
Ricasetron
-
Tedatioxetine
-
Tetracyclic antidepressants (e.g., amoxapine, mianserin, mirtazapine)
-
Thujone
-
Tropanserin
-
Tropisetron
-
Typical antipsychotics (e.g., loxapine)
-
Volatiles/gases (e.g., nitrous oxide, sevoflurane, xenon)
-
Vortioxetine
-
Zacopride
-
Zatosetron
|
|
|
---|
5-HT4 |
|
---|
5-HT5A |
|
---|
5-HT6 |
-
Agonists: Ergolines (e.g., dihydroergocryptine, dihydroergotamine, ergotamine, lisuride, LSD, mesulergine, metergoline, methysergide)
-
Hypidone
-
Serotonin (5-HT)
-
Tryptamines (e.g., 2-Me-5-HT, 5-BT, 5-CT, 5-MT, Bufotenin, E-6801, E-6837, EMD-386088, EMDT, LY-586713, N-Me-5-HT, ST-1936, tryptamine)
-
WAY-181187
-
WAY-208466
|
-
Antagonists: ABT-354
-
Atypical antipsychotics (e.g., aripiprazole, asenapine, clorotepine, clozapine, fluperlapine, iloperidone, olanzapine, tiospirone)
-
AVN-101
-
AVN-211
-
AVN-322
-
AVN-397
-
BGC20-760
-
BVT-5182
-
BVT-74316
-
Cerlapirdine
-
EGIS-12,233
-
GW-742457
-
Idalopirdine
-
Ketanserin
-
Landipirdine
-
Latrepirdine (dimebolin)
-
Masupirdine
-
Metitepine (methiothepin)
-
MS-245
-
PRX-07034
-
Ritanserin
-
Ro 04-6790
-
Ro 63-0563
-
SB-258585
-
SB-271046
-
SB-357134
-
SB-399885
-
SB-742457
-
Tetracyclic antidepressants (e.g., amoxapine, mianserin)
-
Tricyclic antidepressants (e.g., amitriptyline, clomipramine, doxepin, nortriptyline)
-
Typical antipsychotics (e.g., chlorpromazine, loxapine)
|
|
|
---|
5-HT7 |
|
-
Antagonists: Atypical antipsychotics (e.g., amisulpride, aripiprazole, asenapine, brexpiprazole, clorotepine, clozapine, fluperlapine, olanzapine, risperidone, sertindole, tiospirone, ziprasidone, zotepine)
-
Butaclamol
-
DR-4485
-
EGIS-12,233
-
Ergolines (e.g., 2-Br-LSD (BOL-148), amesergide, bromocriptine, cabergoline, dihydroergotamine, ergotamine, LY-53857, LY-215,840, mesulergine, metergoline, methysergide, sergolexole)
-
JNJ-18038683
-
Ketanserin
-
LY-215,840
-
Metitepine (methiothepin)
-
Ritanserin
-
SB-258719
-
SB-258741
-
SB-269970
-
SB-656104
-
SB-656104A
-
SB-691673
-
SLV-313
-
SLV-314
-
Spiperone
-
SSR-181507
-
Tetracyclic antidepressants (e.g., amoxapine, maprotiline, mianserin, mirtazapine)
-
Tricyclic antidepressants (e.g., amitriptyline, clomipramine, imipramine)
-
Typical antipsychotics (e.g., acetophenazine, chlorpromazine, chlorprothixene, fluphenazine, loxapine, pimozide)
-
Vortioxetine
|
|
|
---|
|
---|
|
|